Compile Data Set for Download or QSAR
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Found 6 of ki data for polymerid = 10852
TargetSphingomyelinase C(Bacillus cereus)
Tokushima Bunri University

LigandPNGBDBM248063(SMY-540)
Affinity DataKi:  1.30E+3nM ΔG°:  -8.35kcal/mole IC50:  800nMpH: 7.5 T: 2°CAssay Description:Briefly, Bc-SMase (50 ng/ml) was treated at 37 °C for 60 min with various compounds that were solubilized in dimethylacetoamide. The reaction mix...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSphingomyelinase C(Bacillus cereus)
Tokushima Bunri University

LigandPNGBDBM248063(SMY-540)
Affinity DataKi:  1.30E+3nMAssay Description:Functional potency against Tachykinin receptor 2 (NK2) in rabbit pulmonary artery assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetSphingomyelinase C(Bacillus cereus)
Tokushima Bunri University

LigandPNGBDBM248061(SMY-471)
Affinity DataKi:  2.80E+3nM ΔG°:  -7.87kcal/mole IC50:  900nMpH: 7.5 T: 2°CAssay Description:Briefly, Bc-SMase (50 ng/ml) was treated at 37 °C for 60 min with various compounds that were solubilized in dimethylacetoamide. The reaction mix...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSphingomyelinase C(Bacillus cereus)
Tokushima Bunri University

LigandPNGBDBM248061(SMY-471)
Affinity DataKi:  2.80E+3nMAssay Description:Functional potency against Tachykinin receptor 2 (NK2) in rabbit pulmonary artery assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetSphingomyelinase C(Bacillus cereus)
Tokushima Bunri University

LigandPNGBDBM248057(RY221B-a)
Affinity DataKi:  5.20E+3nM ΔG°:  -7.49kcal/mole IC50:  1.20E+3nMpH: 7.5 T: 2°CAssay Description:Briefly, Bc-SMase (50 ng/ml) was treated at 37 °C for 60 min with various compounds that were solubilized in dimethylacetoamide. The reaction mix...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSphingomyelinase C(Bacillus cereus)
Tokushima Bunri University

LigandPNGBDBM248057(RY221B-a)
Affinity DataKi:  5.20E+3nMAssay Description:Functional potency against Tachykinin receptor 2 (NK2) in rabbit pulmonary artery assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails